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Dr. habil. Agnieszka A. Kaczor

November


Dr. habil. Agnieszka A. Kaczor promoted to a position of associate professor at Medical University of Lublin, Poland.

Dr. habil. Agnieszka A. Kaczor became a member of Molecules Editorial Topic Board. Submissions to Special Issue entitled Targeting Signaling Complexity of GPCRs for the Treatment of CNS Diseases are now invited. Deadline for submission: March 31st, 2021.

3rd award for the best lecture at the COST MuTaLig conference in Izmir, Turkey.

OPUS grant by National Science Center accepted: Novel multi-target ligands of aminergic GPCRs as pharmacological tools to study the pathomechanism of schizophrenia.

OPUS grant by National Sciennce Center in consortium with University of Life Sciences in Lublin (leader) and University of Rzeszow accepted: Dietary polyphenols as thyroid peroxidase (TPO) modulators with multidirectional biological activity - a combined in vitro and in silico investigations.

New articles

Damian Bartuzi, Ewa Kedzierska, Agnieszka A. Kaczor, Helmut Schmidhammer, Dariusz Matosiuk: Novel positive allosteric modulators of µ opioid receptor — insight from in silico and in vivo studies. Int. J. Mol. Sci. 2020, 21, 8463.

Piotr Stepnicki, Magda Kondej, Oliwia Koszla, Justyna Zuk, Agnieszka A. Kaczor: Multi-targeted drug design strategies for the treatment of schizophrenia. Expert Opin. Drug Discov. 2020, in press.

Oliwia Koszla, Magda Kondej, Piotr Stepnicki, Justyna Zuk, Agnieszka A. Kaczor: Neurogenesis and neuroprotection in the hippocampus as the target to treat central nervous system diseases [Polish]. Science and Industry - Lublin Student Meetings, Maria Curie-Sklodowska University, 2020, 109-111.

Justyna Zuk, Oliwia Koszla, Magda Kondej, Piotr Stepnicki, Agnieszka A. Kaczor: Dopaminergic disturbances in the pathomechanism of schizophrenia [Polish]. Science and Industry - Lublin Student Meetings, Maria Curie-Sklodowska University, 2020, 301-304.

Piotr Stepnicki, Magda Kondej, Oliwia Koszla, Justyna Zuk, Anna Kozak, Tomasz M. Wrobel, Agnieszka A. Kaczor: D2AAK2 - a new non-basic ligand of G protein-coupled receptors as a potential antipsychotic [Polish]. Science and Industry - Lublin Student Meetings, Maria Curie-Sklodowska University, 2020, 254-257.

Magda Kondej, Piotr Stepnicki, Oliwia Koszla, Justyna Zuk, Agata Bartyzel, Tomasz M. Wrobel, Andrea G. Silva, Maria I. Loza, Marian Castro, Dariusz Matosiuk, Agnieszka A. Kaczor: Multi-target ligands of aminergic G protein-coupled receptors [Polish]. Science and Industry - Lublin Student Meetings, Maria Curie-Sklodowska University, 2020, 105-108.

Damian Bartuzi, Tomasz M. Wrobel, Agnieszka A. Kaczor, Dariusz Matosiuk: Tuning down the pain – an overview of allosteric modulation of opioid receptors: mechanisms of modulation, allosteric sites, modulator syntheses. Curr. Topics Med. Chem. 2020, in press.

Damian Bartuzi, Agnieszka A. Kaczor, Dariusz Matosiuk: Illuminating the ‘twilight zone’ – advances in difficult protein modeling. Methods Mol. Biol. 2020, in press.

Monika Pitucha, Monika Janeczko, Katarzyna Klimek, Emilia Fornal, Maciej Wos, Anna Pachuta-Stec, Grazyna Ginalska, Agnieszka A. Kaczor: 1,2,4-Triazolin-5-thione derivatives with anticancer activity as CK1γ kinase inhibitors. Bioorg. Chem. 2020, in press.

Agnieszka A. Kaczor, Katarzyna M. Targowska-Duda, Andrea G. Silva. Magda Kondej, Grazyna Biala, Marian Castro: N-(2-hydroxyphenyl)-1-[3-(2-oxo-2,3-dihydro-1H-benzimidazol-1-yl)propyl]piperidine-4-carboxamide (D2AAK4), a multi-target ligand of aminergic GPCRs, as a potential antipsychotic. Biomolecules 2020, 10, 349.

Monika Pitucha, Agnieszka Korga-Plewko, Pawel Kozyra, Mariola Iwan, Agnieszka A. Kaczor: 2,4-Dichlorophenoxyacetic thiosemicarbazides as a new class of compounds against stomach cancer potentially intercalating with DNA. Biomolecules 2020, 10, 296.

Oliwia Koszla, Katarzyna M. Targowska-Duda, Ewa Kedzierska, Agnieszka A. Kaczor: In vitro and in vivo models for the investigation of potential drugs against schizophrenia. Biomolecules 2020, 10, 160.

Justyna Zuk, Damian Bartuzi, Dariusz Matosiuk, Agnieszka A. Kaczor: Preferential coupling of dopamine D2S and D2L receptor isoforms with Gi1and Gi2 proteins - in silico study. Int. J. Mol. Sci. 2020, 21, 436.

Marta Halasa, Damian Bartuzi, Dominika Cieslak, Agnieszka A. Kaczor, Paulina Miziak, Andrzej Stepulak, Dariusz Matosiuk: Role of N-terminus in function and dynamics of Sirtuin 7 – an in silico study. J. Biomol. Struct. Dyn. 2020, 38, 1283-1291.

  
About

Department of Synthesis and Chemical Technology of Pharmaceutical Substances with Computer Modeling Lab, Faculty of Pharmacy with Division of Medical Analytics, Medical University of Lublin, 4A Chodzki St., PL-20093 Lublin, Poland

Google Scholar: Agnieszka A. Kaczor
Researcher ID: A-3744-2015
Orcid: 0000-0001-8679-9623


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